Ke hilinaʻi nei nei kaʻoihanaʻo Parhurcetical i nā pūnaehana Guitika holomua e hoʻomohala i nā lāʻau lapaʻau maikaʻi a me nā lāʻau lapaʻau palekana. Hoʻokahi mea hoʻohui i loaʻa i ka nānā nuiN-boc-glycine isopropylesterster. ^. Ke pāʻani nei kēiaʻano hana maʻamau i kahi hana koʻikoʻi i loko o ka synthesis o nā huahana pharmacetical likeʻole, e hāʻawi ana i nā waiwai hana kūʻokoʻa e hoʻonui ai i nā kaʻina hana hoʻolālā. Ma kēiaʻatikala, eʻimi mākou i nā noi lāʻau lapaʻau o N-BOC-GlyCine isopropylester a no ke aha he mea nui i loko o ka lāʻau lapaʻau hou.
He aha ka mea o n-bol-glycine isopropylester?
ʻO ka n-BOC-Glycine isopropylester kahiʻano chessically hoʻololiʻia o ka glycine, kahi amino acid e lawelaweʻia e like me ka pā hale no nā protein. ʻO ka "n-boc" (thert-birt-butfycarbonyl) hui a me ka nui o ka coropopyl e hoʻonui i nā hui a me ka hana houʻana o ka compound. Hana kēia i ka N-BYC-GlyCine isopropylester i kahi kikowaena koʻikoʻi ma waena o kaʻoihana kūlohelohe ma keʻano o nāʻoihana lāʻau lapaʻau.
ʻO nā noi lāʻau lapaʻau nui o ka N-BOC-GlyCine isopropylesterster
1.ʻO nā synthesis
ʻO kekahi o nā hoʻohana muaʻana o ka N-BOC-Glycine isopropylesters aia i loko o ka synthesis o Peptide. ʻO nā peptides he mau kaulahao pōkoleʻo Amino e pili ana i kahi hana koʻikoʻi i kahi hana koʻikoʻi i nā hana biopical a ua hoʻohanaʻia e like me nā mea lawelawe i hoʻohanaʻia. Mālama ka hui N-BOC i ka hui Amano i ka wā o Synthesis,ʻoiaiʻo ka ISoproyl Estate e hoʻomaʻamaʻa i ka hoʻokumuʻana o nā mea paʻa. Hana kēia i ka n-bol-glycine isopropylester e uku nui no ka hanaʻana i nā pehu i ka maʻemaʻe a me ka hopena.
2.ʻO ke kikowaena lāʻau
Ua hoʻohana nuiʻiaʻo N-BOC-Glycine isopropylesterst e like me kahi waena ma ka synthesis o nāʻano lāʻau lapaʻau likeʻole. Hāʻawi kona mau pūʻulu pale e hana i nā mea kanu e hana i nā hopena koho, e hiki ai ke hana i ka hanaʻana o nā molole paʻakikī. He mea koʻikoʻi kēia i ka hoʻomohalaʻana o nā antibiotics, antiviral, a me nā lāʻau antiniccer.
3.ʻO ka hoʻomohala prodrug
ʻO nā mea hoʻopiʻi i loaʻaʻole i nā mea e hoʻohuli i nā lāʻau lapaʻau ikaika i loko o ke kino. Hiki ke hoʻohanaʻia ka pūʻulu o ka Isopropyl i N-Boltcine isopropyterster He mea pono kēia no nā lāʻau lapaʻau e pono ai e hoʻopili i ka'ōnaehana i hoʻopaʻaʻia a iʻole nā'āpana kiko'ī kiko'ī.
4. E nā mea hoʻonāukiuki Eyzyme
ʻO nā mea hoʻonāukiuki e nā lāʻau lapaʻau he papa o nā lāʻau lapaʻau e pāpā ai i ka hana o nā enzymes kiko'ī, ua hoʻohana pinepineʻia e mālama i nā maʻi a me nā maʻi maʻi maʻi. N-BOC-GAL-Glycine isopropylester e lawelawe i kahi pā hale no ka hoʻopiliʻana i kēia mau inika, e hoʻomaikaʻi i kona hiki ke hana i kahi hiki ke hana i ka hiki ke hana i ka hiki ke hana.
5
ʻO kaʻoiaʻiʻo o ka N-BOC-Glycine isopropylester e hana i kahi pono koʻikoʻi no ka synthes o ke kino maʻamau. Hoʻohanaʻo nā mea noiʻi e hana i nā mea pili i ka novel me nā hopena o nā mea hana ponoʻole.
Loaʻa i ka hoʻohanaʻana i ka hoʻohanaʻana i ka N-Boltcine Glycine Isopropylesterst i nā lāʻau lapaʻau
ʻO ka hoʻohanaʻana o N-BOC-Glycine isopropylesterster i ka hoʻolālāʻana i nā lāʻau lapaʻau e hāʻawi ai i nā mea pono e loaʻa nā pono:
•ʻO ka nui kiʻekiʻe
• Kūpili: Hāʻawi ka hui N-Boc Comb i nā hopena o nā kumumanaʻo i ka hopena o ka pono, e hōʻemi ana i ka hopena o nā hopena i makemakeʻoleʻia.
• Hōʻike:ʻo kāna mau noi noi mai ka synthes synthesis i Prodrugis, e hana ana i kahi mea pono no ka mea noiʻi.
•ʻO ka Scalability: N-BOC-Glycine isopropylester e kūpono no ka noiʻiʻana i nā mea noiʻi liʻiliʻi a me ka hana maʻamau.
Nā pilikia a me nā noʻonoʻo
ʻOiaiʻo N-BOC-GYCINE ISOPROPYLST e hāʻawi i nā pōmaikaʻi nui, e hele ana kona hoʻohanaʻana i nā lāʻau lapaʻau me nā pilikia. No ka manawa, makemakeʻia ka weheʻana o ka hui pale o ka N-Boc. Eia kekahi,ʻo ke kumukūʻai o ke kumukūʻai kiʻekiʻe-ʻo ka hoʻomaʻemaʻe kiʻekiʻe N-bal-glycine isopropylester hiki ke noʻonoʻo no nā noi nui.
ʻOiaiʻo kēia mau pilikia,ʻo ka noiʻiʻana i ka noiʻi a me nā hanaʻenehana e pili ana i kēia mau pilikia, e hana ana i nā kohoʻo N-Boll
ʻO ka wā e hiki mai ana i ka N-BOC-Glycine isopropylesterster i nā lāʻau lapaʻau
Ke hoʻomaka nei ka noiʻana no nā lāʻau lapaʻau a me nā lāʻau lapaʻau maikaʻi, ke hoʻomau nei ka lāʻau lapaʻau ʻO nā holomua ma Synthetic Chemistry a me ke kaʻina hana e hoʻonui ai i kāna mau noi, kūikawā i nā mahina o ka lāʻau lapaʻau pilikino a me nā biologics.
Eia kekahi,ʻo ka uluʻana o ka uluʻana i nā'ōmaʻomaʻo'ōmaʻomaʻo e holo ana i ka hoʻomohalaʻana i nāʻano hana hou aku no ka hoʻopiliʻana a me ka hoʻohanaʻana i n-bol-glycine isopropylester. Ke hoʻololi nei kēia me ke kūpaʻa o kaʻoihana e hōʻemi i konaʻano kūlohelohe i ka wā e hāʻawi ana i nā hana ola.
Hopena
ʻO ka mea nuiʻo N-BOC-Glycine isopylesterster he mea koʻikoʻi i kaʻoihana lāʻau lapaʻau, me nā noi mai ka haku peptide i ka hoʻomohalaʻana. Kona mau waiwai kūʻokoʻa, me nā mea kiʻekiʻe a me ka kūpaʻa, hana i kahi mea hana ikaika loa a me nā mea hana hana a me nā mea hana a me nā mea hana hana a me nā mea hana. Ke hoʻomau nei ka hana i ka hanaʻole, keʻano o ka mea nui o N-BOC-Glycine isopropylester
Ināʻoe e pili ana i ka noiʻi lāʻau lapaʻau a iʻole ka hanaʻana i nā noi a me nā pono o nā lāʻau lapaʻauʻo N-Bolt. Eʻimi pehea e hiki ai i kēiaʻano coundatanile ke hoʻonui i kāu hana a me ka hoʻokeleʻana i keʻano o ka lāʻau lapaʻau.
No nā meaʻike hou aku a me nā'ōlelo akamai, e kipa aku i kā mākou pūnaewele mahttps://www.nvchem.net/e aʻo hou e pili ana i kā mākou huahana a me nā hopena.
Post Time: Mar-17-2025